Atome 2 : Comparative Modeling, Annotation & Complexes Prediction of Study :
PK_HUMAN_I30_2020M9 (2020 - Homo sapiens - Protein Kinase family)

Download : Data.csv | 3D Common Core | 3D Models | DB.fasta


Tab legend :
    Full name of ligand selected in the comparative docking column:

    General color information : Quality: [ Good | Correct | Uncertain ]
QueryStructural Alignment (SA)3D Modeling AnnotationLigands from PDB templatesPredicted Complexes - pKd:[ ‹nMol | ‹μMol | ‹mMol ]




Query Sequence
Filter:
Significants
SA found
Seq Ident. 3D Core
(QMean Score)
Classification code

Binding Site Ligands Found
(Procognate)
Profile Complexes by comparative docking
(ligands from PDB templates)

Targets
for screening


Sort by entries

[Nb of SA]
[Best Ident]
[Best Score]
Main Code
[Name]
[Number]
[Number]
Distribution of CDocking pKd
[Number]
1HCK_HUMAN499 100% 0.68 PF00018 C3_S1597 - (35)20 185 / 214 / 94 217
2TEC_HUMAN515 67% 0.28 PF00018 C2_S1583 - (31)20 183 / 231 / 95 211
3BTK_HUMAN502 100% 0.36 PF00018 C3_S1546 - (31)20 181 / 209 / 106 213
4LYN_HUMAN485 100% 0.48 PF00018 C3_S1574 - (30)20 180 / 198 / 102 188
5BLK_HUMAN508 75% 0.43 PF00018 C3_S1597 - (31)20 179 / 214 / 109 209
6LCK_HUMAN484 100% 0.56 PF00018 C2_S1570 - (32)20 170 / 203 / 105 214
7BMX_HUMAN513 98% 0.26 PF00018 C1_S1586 - (32)20 167 / 234 / 103 198
8ABL1_HUMAN507 100% 0.32 PF00018 C4_S1596 - (30)20 163 / 224 / 116 131
9SRMS_HUMAN477 56% 0.42 PF00018 C3_S1576 - (31)20 161 / 213 / 96 183
10TXK_HUMAN513 66% 0.27 PF00018 C1_S1572 - (31)20 160 / 225 / 124 219
11ABL2_HUMAN504 100% 0.33 PF00018 C5_S1582 - (32)20 157 / 225 / 120 130
12FGFR3_HUMAN466 98% 0.22 PF00018 C4_S1584 - (69)20 154 / 196 / 105 157
13DDR1_HUMAN491 100% 0.20 PF00018 C1_S1594 - (75)20 151 / 207 / 128 107
14FGFR1_HUMAN448 100% 0.22 PF00018 C6_S1565 - (70)20 151 / 186 / 98 153
15FYN_HUMAN452 85% 0.67 PF00018 C4_S1522 - (22)20 149 / 191 / 91 182
16FGR_HUMAN452 80% 0.53 PF00018 C1_S1528 - (22)20 147 / 205 / 80 184
17YES_HUMAN454 90% 0.70 PF00018 C2_S1531 - (26)20 147 / 199 / 83 178
18EPHB1_HUMAN470 100% 0.17 PF00018 C2_S1517 - (42)20 146 / 193 / 123 156
19EPHA2_HUMAN479 100% 0.18 PF00018 C5_S1528 - (45)20 145 / 191 / 136 164
20FRK_HUMAN411 61% 0.46 PF00018 C3_S1455 - (26)20 141 / 182 / 80 166
21DDR2_HUMAN494 100% 0.17 PF00018 C1_S1548 - (80)20 140 / 204 / 133 108
22EPHB4_HUMAN489 100% 0.18 PF00018 C2_S1519 - (45)20 139 / 199 / 138 155
23PTK6_HUMAN499 99% 0.32 PF00018 C4_S1568 - (65)20 138 / 217 / 134 171
24EPHB2_HUMAN469 100% 0.15 PF00018 C1_S1509 - (42)20 138 / 185 / 134 149
25EPHA5_HUMAN468 88% 0.17 PF00018 C2_S1496 - (45)20 135 / 189 / 129 154
26EPHA1_HUMAN485 62% 0.18 PF00018 C4_S1532 - (44)20 134 / 191 / 149 158
27EPHB3_HUMAN455 99% 0.17 PF00018 C3_S1496 - (43)20 134 / 183 / 130 154
28CSK_HUMAN513 100% 0.59 PF00018 C2_S1608 - (32)20 133 / 220 / 145 200
29EPHA3_HUMAN462 99% 0.18 PF00018 C1_S1486 - (45)20 132 / 181 / 133 147
30EPHA4_HUMAN464 99% 0.21 PF00018 C2_S1511 - (45)20 130 / 183 / 139 166
31FER_HUMAN486 67% 0.27 PF00018 C2_S1564 - (40)20 129 / 208 / 138 140
32SRC_HUMAN320 100% 0.72 PF00018 C2_S1353 - (19)20 124 / 119 / 57 132
33FAK2_HUMAN414 100% 0.31 PF00018 C3_S1480 - (57)20 123 / 189 / 97 111
34MERTK_HUMAN443 100% 0.17 PF00018 C3_S1577 - (63)20 117 / 198 / 117 117
35UFO_HUMAN422 100% 0.17 PF00018 C5_S1548 - (59)20 115 / 165 / 128 129
36ERBB4_HUMAN396 100% 0.13 PF00018 C5_S1435 - (61)183 113 / 194 / 84 131
37TYRO3_HUMAN378 98% 0.14 PF00018 C5_S1474 - (39)20 113 / 169 / 83 107
38MK14_HUMAN453 100% 0.78 PF00069 C1_S1541 - (40)20 110 / 210 / 110 307
39MATK_HUMAN515 59% 0.47 PF00018 C2_S1599 - (62)20 109 / 188 / 207 156
40MK11_HUMAN449 100% 0.48 PF00069 C1_S1574 - (42)20 108 / 213 / 112 302
41EPHA6_HUMAN462 74% 0.17 PF00018 C3_S1491 - (36)20 103 / 194 / 155 121
42TNK1_HUMAN358 49% 0.27 PF00018 C1_S1407 - (63)20 99 / 157 / 88 86
43MK09_HUMAN444 98% 0.39 PF00069 C1_S1520 - (31)20 98 / 231 / 105 278
44ALK_HUMAN391 100% 0.10 PF00018 C2_S1459 - (57)20 98 / 176 / 99 94
45ACK1_HUMAN365 100% 0.16 PF00018 C5_S1424 - (62)20 98 / 147 / 111 58
46FAK1_HUMAN389 100% 0.31 PF00018 C2_S1430 - (38)20 97 / 171 / 108 109
47KIT_HUMAN490 99% 0.16 PF00018 C4_S1605 - (61)20 97 / 170 / 201 60
48JAK2_HUMAN437 99% 0.22 PF00018 C1_S1490 - (20)20 95 / 266 / 73 145
49MK10_HUMAN446 100% 0.41 PF00069 C2_S1545 - (29)20 93 / 227 / 113 276
50BRAF_HUMAN176 100% 0.22 PF02196 C3_S1209 - (6)20 91 / 51 / 15 67

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